Difference between revisions of "Template:Estrogen receptor modulators"

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{{Navbox
 
{{Navbox
−
| name  = Estrogenics
+
| name  = Estrogen receptor modulators
−
| title = [[Estrogen]]ics
+
| title = [[Estrogen receptor]] [[receptor modulator|modulator]]s
−
| listclass = hlist
+
| bodyclass = hlist
 
| state = {{{state<includeonly>|collapsed</includeonly>}}}
 
| state = {{{state<includeonly>|collapsed</includeonly>}}}
−
| groupstyle = text-align:center;
+
| groupstyle = text-align:center;  
  
−
   | group1 = [[Receptor (biochemistry)|Receptor]]<br /><small>([[Ligand (biochemistry)|ligands]])</small>
+
   | group1 = {{abbrlink|ER|Estrogen receptor}}
−
   |  list1 = {{Navbox subgroup
+
   | list1 = {{Navbox|subgroup
−
   | groupstyle = text-align:center;
+
   | groupstyle = text-align:center
 +
  | groupwidth = 6em;
  
−
     | group1 = [[Estrogen receptor|ER]] ([[Estrogen receptor alpha|α]], [[Estrogen receptor beta|β]])
+
     | group1 = Agonists
−
     | list1 = {{Navbox subgroup
+
     | list1 =
−
    | groupstyle = text-align:center;
+
* ''Steroidal:'' [[2-Hydroxyestradiol]]
−
 
+
* [[2-Hydroxyestrone]]
−
      | group1 = Agonists
+
* [[3-Methyl-19-methyleneandrosta-3,5-dien-17β-ol]]
−
      | list1 =
 
−
* [[(R)-DPN]]
 
−
* [[(S)-DPN]]
 
−
* [[(R,R)-Tetrahydrochrysene|(R,R)-THC]]
 
−
* [[(S,S)-Tetrahydrochrysene|(S,S)-THC]]
 
−
* [[2,8-Dihydroxyhexahydrochrysene|2,8-DHHHC]]
 
 
* [[3α-Androstanediol]]
 
* [[3α-Androstanediol]]
−
* [[3β-Androstanediol]]
+
* [[3α,5α-Dihydrolevonorgestrel]]
 +
* [[3β,5α-Dihydrolevonorgestrel]]
 
* [[3α-Hydroxytibolone]]
 
* [[3α-Hydroxytibolone]]
 
* [[3β-Hydroxytibolone]]
 
* [[3β-Hydroxytibolone]]
−
* [[7-Oxo-DHEA]]
+
* [[3β-Androstanediol]]
 +
* [[4-Androstenediol]]
 +
* [[4-Androstenedione]]
 +
* [[4-Fluoroestradiol]]
 +
* [[4-Hydroxyestradiol]]
 +
* [[4-Hydroxyestrone]]
 +
* [[4-Methoxyestradiol]]
 +
* [[4-Methoxyestrone]]
 +
* [[5-Androstenediol]]
 +
* [[7-Keto-DHEA|7-Oxo-DHEA]]
 
* [[7α-Hydroxy-DHEA]]
 
* [[7α-Hydroxy-DHEA]]
 +
* [[7α-Methylestradiol]]
 
* [[7β-Hydroxyepiandrosterone]]
 
* [[7β-Hydroxyepiandrosterone]]
−
* [[8β-VE2|8β-VE<sub>2</sub>]]
+
* [[8,9-Dehydroestradiol]]
−
* [[16-Hydroxydehydroepiandrosterone|16α-Hydroxy-DHEA]]
+
* [[8,9-Dehydroestrone]]
 +
* [[8β-VE2]]
 +
* [[10β,17β-Dihydroxyestra-1,4-dien-3-one|10β,17β-Dihydroxyestra-1,4-dien-3-one (DHED)]]
 +
* [[11β-Chloromethylestradiol]]
 +
* [[11β-Methoxyestradiol]]
 +
* [[15α-Hydroxyestradiol]]
 +
* [[16-Ketoestradiol]]
 +
* [[16-Ketoestrone]]
 +
* [[16α-Fluoroestradiol]]
 +
* [[16α-Hydroxy-DHEA]]
 
* [[16α-Hydroxyestrone]]
 
* [[16α-Hydroxyestrone]]
−
* [[16α-Iodo-E2|16α-IE<sub>2</sub>]]
+
* [[16α-Iodoestradiol]]
−
* [[16α-LE2|16α-LE<sub>2</sub> (Cpd1471)]]
+
* [[16α-LE2]]
−
* [[Δ4-Androstenedione|Δ<sup>4</sup>-Androstenedione]]
+
* [[16β-Hydroxyestrone]]
−
* [[Δ5-Androstenediol|Δ<sup>5</sup>-Androstenediol]]
+
* [[16β,17α-Epiestriol|16β,17α-Epiestriol (16β-hydroxy-17α-estradiol)]]
−
* [[Alfatradiol|17α-Estradiol (alfatradiol)]]
+
* [[17α-Estradiol]] ([[alfatradiol]])
−
* [[Estradiol|17β-Estradiol (estradiol)]]
+
* [[17α-Dihydroequilenin]]
 +
* [[17α-Dihydroequilin]]
 +
* [[17α-Epiestriol|17α-Epiestriol (16α-hydroxy-17α-estradiol)]]
 +
* [[17α-Ethynyl-3α-androstanediol]]
 +
* [[17α-Ethynyl-3β-androstanediol]]
 +
* [[17β-Dihydroequilenin]]
 +
* [[17β-Dihydroequilin]]
 +
* [[17β-Methyl-17α-dihydroequilenin]]
 +
* [[Abiraterone]]
 +
* [[Abiraterone acetate]]
 
* [[Alestramustine]]
 
* [[Alestramustine]]
 
* [[Almestrone]]
 
* [[Almestrone]]
−
* [[Anabolic steroid]]s ([[prodrug]]s; e.g., [[testosterone]], [[metandienone|metandienone (methandrostenolone)]], others)
+
* [[Anabolic steroid]]s (e.g., [[testosterone]] and [[List of androgen esters#Testosterone esters|ester]]s, [[methyltestosterone]], [[metandienone|metandienone (methandrostenolone)]], [[nandrolone]] and [[List of androgen esters#Nandrolone esters|ester]]s, many others; via estrogenic metabolites)
−
* [[Anethole]]
 
−
* [[Anol (drug)|Anol]]
 
 
* [[Atrimustine]]
 
* [[Atrimustine]]
−
* [[Benzestrol]]
+
* [[Bolandiol]]
−
* [[Bifluranol]]
+
* [[Bolandiol dipropionate]]
−
* [[Bisdehydrodoisynolic acid]]
+
* [[Butolame]]
−
* [[Carbestrol]]
+
* [[Clomestrone]]
−
* [[Chalconoid]]s (e.g., [[isoliquiritigenin]], [[phloretin]], [[phlorizin|phlorizin (phloridzin)]], [[wedelolactone]])
 
 
* [[Cloxestradiol]]
 
* [[Cloxestradiol]]
−
* [[Conjugated equine estrogen]]s (e.g., [[sodium equilin sulfate]], [[sodium equilenin sulfate]])
+
** [[Cloxestradiol acetate]]
−
* [[Coumestan]]s (e.g., [[coumestrol]], [[psoralidin]])
+
* [[Conjugated estriol]]
−
* [[DBE (drug)|DBE]]
+
* [[Conjugated estrogens]]
 +
* [[Cyclodiol]]
 +
* [[Cyclotriol]]
 
* [[Dehydroepiandrosterone|DHEA]]
 
* [[Dehydroepiandrosterone|DHEA]]
 
* [[Dehydroepiandrosterone|DHEA-S]]
 
* [[Dehydroepiandrosterone|DHEA-S]]
−
* [[Deoxymiroestrol]]
+
* [[ent-Estradiol|''ent''-Estradiol]]
−
* [[Dianethole]]
+
* [[Epiestriol|Epiestriol (16β-epiestriol, 16β-hydroxy-17β-estradiol)]]
−
* [[Dianol]]
 
−
* [[Diarylpropionitrile]]
 
−
* [[Dieldrin]]
 
−
* [[Dienestrol]]
 
−
* [[Dienestrol acetate]]
 
−
* [[Diethylstilbestrol]]
 
−
* [[Diethylstilbestrol dipropionate]]
 
−
* [[Diosgenin]]
 
−
* [[Doisynoestrol|Doisynoestrol (fenocycline)]]
 
−
* [[Doisynolic acid]]
 
−
* [[DY-131|DY-131 (GSK-9089)]]
 
−
* [[Endosulfan]]
 
−
* [[Epiestriol]]
 
 
* [[Epimestrol]]
 
* [[Epimestrol]]
−
* [[ERB-196|ERB-196 (WAY-202196)]]
+
* [[Equilenin]]
−
* [[Esterified estrogen]]s (e.g., [[estrone sulfate]], [[equilin sulfate]], [[equilenin sulfate]])
+
* [[Equilin]]
 +
* [[ERA-63|ERA-63 (ORG-37663)]]
 +
* [[Esterified estrogens]]
 
* [[Estetrol]]
 
* [[Estetrol]]
−
* [[Estradiol benzoate]]
+
* [[Estradiol]]
−
* [[Estradiol butyrylacetate]]
+
** [[List of estrogen esters#Estradiol esters|Estradiol esters]]
−
* [[Estradiol cypionate]]
+
** [[Lipoidal estradiol]]
−
* [[Estradiol dienanthate]]
+
** [[Polyestradiol phosphate]]
−
* [[Estradiol dipropionate]]
 
−
* [[Estradiol diundecylate]]
 
−
* [[Estradiol diundecylenate]]
 
−
* [[Estradiol enanthate]]
 
−
* [[Estradiol furoate]]
 
−
* [[Estradiol hemihydrate]]
 
−
* [[Estradiol hemisuccinate]]
 
−
* [[Estradiol hexahydrobenzoate]]
 
−
* [[Estradiol monopropionate]]
 
−
* [[Estradiol palmitate]]
 
−
* [[Estradiol pivalate]]
 
−
* [[Estradiol propoxyphenylpropionate]]
 
−
* [[Estradiol stearate]]
 
−
* [[Estradiol succinate]]
 
−
* [[Estradiol undecylate]]
 
−
* [[Estradiol valerate]]
 
 
* [[Estramustine]]
 
* [[Estramustine]]
 
* [[Estramustine phosphate]]
 
* [[Estramustine phosphate]]
Line 98: Line 94:
 
* [[Estrazinol]]
 
* [[Estrazinol]]
 
* [[Estriol]]
 
* [[Estriol]]
−
* [[Estriol succinate]]
+
** [[List of estrogen esters#Estriol esters|Estriol esters]]
−
* [[Estriol tripropionate]]
+
** [[Polyestriol phosphate]]
 
* [[Estrofurate]]
 
* [[Estrofurate]]
 +
* [[Estrogenic substances]]
 
* [[Estromustine]]
 
* [[Estromustine]]
 
* [[Estrone]]
 
* [[Estrone]]
−
* [[Estrone acetate]]
+
** [[List of estrogen esters#Estrone esters|Estrone esters]]
−
* [[Estrone cyanate]]
+
** [[Estrone methyl ether]]
−
* [[Estrone sulfate]]
+
** [[Estropipate]]
−
* [[Estrone tetraacetylglucoside]]
 
−
* [[Estropipate]]
 
−
* [[Estropronicate]]
 
 
* [[Etamestrol|Etamestrol (eptamestrol)]]
 
* [[Etamestrol|Etamestrol (eptamestrol)]]
−
* [[Ethinyl estradiol]]
+
* [[Ethinylandrostenediol]]
−
* [[Ethinyl estradiol 3-isopropylsulfonate]]
+
** [[Ethandrostate]]
 +
* [[Ethinylestradiol]]
 +
** [[Ethinylestradiol 3-benzoate]]
 +
** [[Ethinylestradiol sulfonate]]
 +
* [[Ethinylestriol]]
 +
* [[Ethylestradiol]]
 +
* [[Etynodiol]]
 
* [[Etynodiol diacetate]]
 
* [[Etynodiol diacetate]]
−
* [[Fenarimol]]
+
* [[Hexolame]]
−
* [[Fenestrel]]
+
* [[Hippulin]]
−
* [[2-Chloro-3'-fluoro-3,4'-dihydroxy-(1,1-biphenyl)-4-carboxaldehyde oxime|FERb 033]]
 
−
* [[Flavonoid]]s (incl. [[7,8-Dihydroxyflavone|7,8-DHF]], [[8-Prenylnaringenin|8-prenylnaringenin]], [[apigenin]], [[baicalein]], [[baicalin]], [[calycosin]], [[catechin]], [[daidzein]], [[daidzin]], [[epicatechin gallate|ECG]], [[epigallocatechin gallate|EGCG]], [[epicatechin]], [[equol]], [[formononetin]], [[glabrene]], [[glabridin]], [[genistein]], [[genistin]], [[glycitein]], [[kaempferol]], [[liquiritigenin]], [[mirificin]], [[myricetin]], [[naringenin]], [[pinocembrin]], [[prunetin]], [[puerarin]], [[quercetin]], [[tectoridin]], [[tectorigenin]])
 
−
* [[Fosfestrol]]
 
−
* [[Furostilbestrol]]
 
−
* [[GSK-4716]]
 
−
* [[Hexestrol]]
 
−
* [[Hexestrol diacetate]]
 
−
* [[Hexestrol dicaprylate]]
 
−
* [[Hexestrol diphosphate]]
 
−
* [[Hexestrol dipropionate]]
 
 
* [[Hydroxyestrone diacetate]]
 
* [[Hydroxyestrone diacetate]]
−
* [[Lavender oil]]
+
* [[Lynestrenol]]
−
* [[Lignan]]s (e.g., [[enterodiol]], [[enterolactone]])
+
* [[Lynestrenol phenylpropionate]]
 
* [[Mestranol]]
 
* [[Mestranol]]
−
* [[Metalloestrogen]]s (e.g., [[cadmium]])
 
−
* [[Methallenestril]]
 
−
* [[Methestrol]]
 
−
* [[Methestrol dipropionate]]
 
−
* [[Methiocarb]]
 
 
* [[Methylestradiol]]
 
* [[Methylestradiol]]
−
* [[Miroestrol]]
 
 
* [[Moxestrol]]
 
* [[Moxestrol]]
 +
* [[Mytatrienediol]]
 
* [[Nilestriol]]
 
* [[Nilestriol]]
 +
* [[Norethisterone]]
 
* [[Noretynodrel]]
 
* [[Noretynodrel]]
 
* [[Orestrate]]
 
* [[Orestrate]]
 +
* [[Pentolame]]
 +
* [[Prodiame]]
 +
* [[Prolame]]
 +
* [[Promestriene]]
 +
* [[RU-16117]]
 +
* [[Quinestradol]]
 +
* [[Quinestrol]]
 +
* [[Tibolone]]
 +
 +
* ''Nonsteroidal:'' [[(R,R)-Tetrahydrochrysene|(R,R)-THC]]
 +
* [[(S,S)-Tetrahydrochrysene|(S,S)-THC]]
 +
* [[2,8-Dihydroxyhexahydrochrysene|2,8-DHHHC]]
 +
* [[β-LGND1]]
 +
* [[β-LGND2|β-LGND2 (GTx-878)]]
 +
* [[AC-186]]
 +
* [[Allenestrol]]
 +
* [[Allenolic acid]]
 +
* [[Benzestrol]]
 +
* [[Bifluranol]]
 +
* [[Bisdehydrodoisynolic acid]]
 +
* [[Butestrol]]
 +
* [[Carbestrol]]
 +
* [[D-15414]]
 +
* [[DCW234]]
 +
* [[Diarylpropionitrile]]
 +
* [[Dienestrol]]
 +
** [[Dienestrol diacetate]]
 +
* [[Diethylstilbestrol]]
 +
** [[List of estrogen esters#Diethylstilbestrol esters|Diethylstilbestrol esters]]
 +
* [[Dimestrol|Dimestrol (dianisylhexene)]]
 +
* [[Dimethylstilbestrol]]
 +
* [[Doisynoestrol|Doisynoestrol (fenocycline)]]
 +
* [[Doisynolic acid]]
 +
* [[Efavirenz]]
 +
* [[ERB-196|ERB-196 (WAY-202196)]]
 +
* [[Erteberel|Erteberel (SERBA-1, LY-500307)]]
 +
* [[Estrobin|Estrobin (DBE)]]
 +
* [[Fenestrel]]
 +
* [[FERb 033]]
 +
* [[Fosfestrol|Fosfestrol (diethylstilbestrol diphosphate)]]
 +
* [[Furostilbestrol|Furostilbestrol (diethylstilbestrol difuroate)]]
 +
* [[GTx-758]]
 +
* [[Hexestrol]]
 +
** [[List of estrogen esters#Hexestrol esters|Hexestrol esters]]
 +
* [[ICI-85966|ICI-85966 (Stilbostat)]]
 +
* [[M2613]]
 +
* [[meso-Butestrol|''meso''-Butestrol]]
 +
* [[meso-Hexestrol|''meso''-Hexestrol]]
 +
* [[Mestilbol]]
 +
* [[Methallenestril]]
 +
* [[Methestrol]]
 +
* [[Methestrol dipropionate]]
 
* [[Paroxypropione]]
 
* [[Paroxypropione]]
−
* [[Phytosterol]]s (e.g., [[β-sitosterol]], [[campesterol]], [[stigmasterol]])
+
* [[Pentafluranol]]
−
* [[Polyestradiol phosphate]]
+
* [[Phenestrol]]
 
* [[Prinaberel|Prinaberel (ERB-041, WAY-202041)]]
 
* [[Prinaberel|Prinaberel (ERB-041, WAY-202041)]]
 
* [[Propylpyrazoletriol]]
 
* [[Propylpyrazoletriol]]
−
* [[Promestriene]]
 
−
* [[Resorcylic acid lactone]]s (e.g., [[zearalanone]], [[zearalenol]], [[zearalenone]], [[zeranol|zeranal (zearalanol)]])
 
 
* [[Quadrosilan]]
 
* [[Quadrosilan]]
−
* [[Quinestradol]]
+
* [[SC-3296]]
−
* [[Quinestrol]]
+
* [[SC-4289]]
 +
* [[SERBA-2]]
 
* [[SKF-82,958]]
 
* [[SKF-82,958]]
−
* [[Stilbenoid]]s (e.g., [[resveratrol]])
+
* [[Terfluranol]]
 +
* [[Triphenylbromoethylene]]
 +
* [[Triphenylchloroethylene]]
 +
* [[Triphenyliodoethylene]]
 +
* [[Triphenylmethylethylene|Triphenylmethylethylene (triphenylpropene)]]
 +
* [[WAY-166818]]
 +
* [[WAY-169916]]
 +
* [[WAY-200070]]
 +
* [[WAY-204688|WAY-204688 (SIM-688)]]
 +
* [[WAY-214156]]
 +
 
 +
* ''Unknown/unsorted:'' [[ERB-26]]<!--Selective ERβ agonist; active enantiomer of ERB-79-->
 +
* [[ERA-45]]<!--Selective ERα agonist-->
 +
* [[ERB-79]]<!--Selective ERβ agonist-->
 +
* [[ZK-283197]]<!--Selective ERβ agonist-->
 +
 
 +
* ''Xenoestrogens:'' [[Anise]]-related (e.g., [[anethole]], [[anol]], [[dianethole]], [[dianol]], [[photoanethole]])
 +
* [[Chalconoid]]s (e.g., [[isoliquiritigenin]], [[phloretin]], [[phlorizin|phlorizin (phloridzin)]], [[wedelolactone]])
 +
* [[Coumestan]]s (e.g., [[coumestrol]], [[psoralidin]])
 +
* [[Flavonoid]]s (incl. [[7,8-Dihydroxyflavone|7,8-DHF]], [[8-Prenylnaringenin|8-prenylnaringenin]], [[apigenin]], [[baicalein]], [[baicalin]], [[biochanin A]], [[calycosin]], [[catechin]], [[daidzein]], [[daidzin]], [[epicatechin gallate|ECG]], [[epigallocatechin gallate|EGCG]], [[epicatechin]], [[equol]], [[formononetin]], [[glabrene]], [[glabridin]], [[genistein]], [[genistin]], [[glycitein]], [[kaempferol]], [[liquiritigenin]], [[mirificin]], [[myricetin]], [[naringenin]], [[penduletin]], [[pinocembrin]], [[prunetin]], [[puerarin]], [[quercetin]], [[tectoridin]], [[tectorigenin]])
 +
* [[Lavender oil]]
 +
* [[Lignan]]s (e.g., [[enterodiol]], [[enterolactone]], [[nyasol|nyasol (''cis''-hinokiresinol)]])
 +
* [[Metalloestrogen]]s (e.g., [[cadmium]])
 +
* [[Pesticide]]s (e.g., [[alternariol]], [[dieldrin]], [[endosulfan]], [[fenarimol]], [[HPTE]], [[methiocarb]], [[methoxychlor]], [[triclocarban]], [[triclosan]])
 +
* [[Phytosteroid]]s (e.g., [[digitoxin]] ([[digitalis]]), [[diosgenin]], [[guggulsterone]])
 +
* [[Phytosterol]]s (e.g., [[β-sitosterol]], [[campesterol]], [[stigmasterol]])
 +
* [[Resorcylic acid lactone]]s (e.g., [[zearalanone]], [[α-zearalenol]], [[β-zearalenol]], [[zearalenone]], [[zeranol|zeranol (α-zearalanol)]], [[taleranol|taleranol (teranol, β-zearalanol)]])
 +
* [[Steroid]]-like (e.g., [[deoxymiroestrol]], [[miroestrol]])
 +
* [[Stilbenoid]]s (e.g., [[resveratrol]], [[rhaponticin]])
 
* [[Synthetic xenoestrogen]]s (e.g., [[alkylphenol]]s, [[bisphenol]]s (e.g., [[bisphenol A|BPA]], [[bisphenol F|BPF]], [[bisphenol S|BPS]]), [[dichlorodiphenyltrichloroethane|DDT]], [[paraben]]s, [[polybrominated biphenyl|PBBs]], [[4-hydroxybenzoic acid|PHBA]], [[phthalate]]s, [[polychlorinated biphenyl|PCBs]])
 
* [[Synthetic xenoestrogen]]s (e.g., [[alkylphenol]]s, [[bisphenol]]s (e.g., [[bisphenol A|BPA]], [[bisphenol F|BPF]], [[bisphenol S|BPS]]), [[dichlorodiphenyltrichloroethane|DDT]], [[paraben]]s, [[polybrominated biphenyl|PBBs]], [[4-hydroxybenzoic acid|PHBA]], [[phthalate]]s, [[polychlorinated biphenyl|PCBs]])
−
* [[WAY-166818]]
+
* Others (e.g., [[agnuside]], [[rotundifuran]])
−
* [[WAY-200070]]<!--7-Bromo-2-(4-hydroxyphenyl)-1,3-benzoxazol-5-ol-->
 
  
−
      | group2 = Mixed ([[Selective estrogen receptor modulator|SERMs]])
+
    | group2 = Mixed<br />({{abbrlink|SERMs|Selective estrogen receptor modulators}})
−
      | list2 =
+
    | list2 =
−
* [[2-Hydroxyestrone]]
+
* [[2-Phenylbenzofuran]]
 +
* [[2-Phenylbenzothiophene]]
 +
* [[4'-Hydroxynorendoxifen]]
 
* [[27-Hydroxycholesterol]]
 
* [[27-Hydroxycholesterol]]
 +
* [[Acefluranol]]
 
* [[Acolbifene]]
 
* [[Acolbifene]]
 
* [[Afimoxifene]]
 
* [[Afimoxifene]]
 +
* [[Anordiol]]
 
* [[Anordrin]]
 
* [[Anordrin]]
−
* [[Anordriol]]
 
 
* [[Arzoxifene]]
 
* [[Arzoxifene]]
 
* [[Bazedoxifene]]
 
* [[Bazedoxifene]]
 +
* [[Brilanestrant]]
 
* [[Broparestrol]]
 
* [[Broparestrol]]
 
* [[Chlorotrianisene]]
 
* [[Chlorotrianisene]]
 
* [[Clomifene]]
 
* [[Clomifene]]
 
* [[Clomifenoxide]]
 
* [[Clomifenoxide]]
 +
* [[CN-55945-27]]
 
* [[Cyclofenil]]
 
* [[Cyclofenil]]
 +
* [[D-15413]]
 +
* [[Desmethylchlorotrianisene]]
 
* [[Droloxifene]]
 
* [[Droloxifene]]
 +
* [[Elacestrant]]
 
* [[Enclomifene]]
 
* [[Enclomifene]]
 
* [[Endoxifen]]
 
* [[Endoxifen]]
 +
* [[Etacstil|Etacstil (GW-5638, DPC-974)]]
 
* [[Ethamoxytriphetol|Ethamoxytriphetol (MER-25)]]
 
* [[Ethamoxytriphetol|Ethamoxytriphetol (MER-25)]]
 
* [[Femarelle]]
 
* [[Femarelle]]
 
* [[Fispemifene]]
 
* [[Fispemifene]]
−
* [[3-(4-(1,2-Diphenylbut-1-enyl)phenyl)acrylic acid|GW5638]]
+
* [[GW-7604]]
 +
* [[ICI-55548]]<!--N--desmethyltamoxifen-->
 
* [[Idoxifene]]
 
* [[Idoxifene]]
 
* [[Lasofoxifene]]
 
* [[Lasofoxifene]]
 
* [[Levormeloxifene]]
 
* [[Levormeloxifene]]
 +
* [[LN-1643]]
 +
* [[LN-2299]]
 +
* [[LY-117018]]<!--63676-25-5; benzothiophene derivative-->
 
* [[Menerba]]
 
* [[Menerba]]
−
* [[Mepitiostane]]
 
 
* [[Miproxifene]]
 
* [[Miproxifene]]
 +
* [[Miproxifene phosphate]]
 +
* [[MRL-37]]
 
* [[Nafoxidine]]
 
* [[Nafoxidine]]
 
* [[Nitromifene]]
 
* [[Nitromifene]]
 +
* [[NNC 45-0095]]
 +
* [[NNC 45-0320]]
 +
* [[NNC 45-0781]]
 +
* [[NNC 45-1506]]
 
* [[Ormeloxifene]]
 
* [[Ormeloxifene]]
 
* [[Ospemifene]]
 
* [[Ospemifene]]
 
* [[Panomifene]]
 
* [[Panomifene]]
−
* [[Phenytoin]]
 
 
* [[Pipendoxifene]]
 
* [[Pipendoxifene]]
 +
* [[Promensil]]
 
* [[Raloxifene]]
 
* [[Raloxifene]]
−
* [[2E-3-(4-((Z)-4-Chloro-1,2-diphenylbut-1-enyl)phenyl)acrylic acid|SS1010]]
+
* [[Rimostil|Rimostil (P-081)]]
−
* [[Sivifene]]
+
* [[Spironolactone]]
 +
* [[SS1010]]<!--2E-3-(4-((Z)-4-Chloro-1,2-diphenylbut-1-enyl)phenyl)acrylic acid-->
 
* [[Tamoxifen]]
 
* [[Tamoxifen]]
−
* [[(7R,8S,9S,13R,14S,17R)-17-(2-(4-((Diethylamino)methyl)-2-methoxyphenoxy)ethyl)-7,13-dimethyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta(a)phenanthren-3-ol 2-hydroxypropane-1,2,3-tricarboxylate|TAS-108]]
+
* [[TAS-108|TAS-108 (SR-16234)]]
−
* [[Tesmilifene]]
 
−
* [[Tibolone]]
 
 
* [[Toremifene]]
 
* [[Toremifene]]
 
* [[Trioxifene]]
 
* [[Trioxifene]]
−
* [[(6-Hydroxy-2-(4-hydroxyphenyl)benzo(b)thien-3-yl)-(4-(4-(1-methylethyl)-1-piperazinyl)phenyl)methanone|Y-134]]
+
* [[TZE-5323]]
 +
* [[U-11555A]]
 +
* [[U-11634]]
 +
* [[Y-134]]<!--(6-Hydroxy-2-(4-hydroxyphenyl)benzo(b)thien-3-yl)-(4-(4-(1-methylethyl)-1-piperazinyl)phenyl)methanone-->
 
* [[Zindoxifene]]
 
* [[Zindoxifene]]
 
* [[Zuclomifene]]
 
* [[Zuclomifene]]
  
−
      | group3 = Antagonists
+
    | group3 = Antagonists
−
      | list3 =
+
    | list3 =
 
* [[(R,R)-Tetrahydrochrysene|(R,R)-THC]]
 
* [[(R,R)-Tetrahydrochrysene|(R,R)-THC]]
−
* [[Fulvestrant]]
+
* [[7β-Hydroxy-DHEA]]
 +
* [[Chloroindazole]]
 +
* [[Cytestrol acetate]]
 +
* [[EM-800|EM-800 (SCH-57050)]]
 +
* [[Epitiostanol]]
 +
* [[ERA-90]]<!--Selective ERα antagonist-->
 +
* [[ERB-88]]<!--Selective ERβ antagonist-->
 +
* [[Fulvestrant|Fulvestrant (ICI-182780)]]
 +
* [[Glyceollin]]s ([[Glyceollin I|I]], [[Glyceollin II|II]], [[Glyceollin III|III]], [[Glyceollin IV|IV]])
 
* [[ICI-164384]]
 
* [[ICI-164384]]
 +
* [[MDL-101906]]
 +
* [[Mepitiostane]]
 +
* [[Methylepitiostanol]]
 
* [[Methylpiperidinopyrazole]]
 
* [[Methylpiperidinopyrazole]]
 
* [[MIBE]]
 
* [[MIBE]]
 +
* [[Oxabicycloheptene sulfonate]]
 +
* [[Phenytoin]]
 
* [[PHTPP]]
 
* [[PHTPP]]
 
* [[Prochloraz]]
 
* [[Prochloraz]]
 +
* [[RU-39411]]
 
* [[RU-58668]]
 
* [[RU-58668]]
 
* [[SS1020]]
 
* [[SS1020]]
−
* [[XCT-790]]
+
* [[TAS-108|TAS-108 (SR-16234)]]
 +
* [[ZB716]]<!--Fulvestrant-3 boronic acid-->
 
* [[ZK-164015]]
 
* [[ZK-164015]]
 
* [[ZK-191703]]
 
* [[ZK-191703]]
  
−
    }}
+
* ''Coregulator-binding modulators:'' [[ERX-11]]
  
−
    | group2 = '''[[G protein-coupled estrogen receptor 1|GPER]]'''
+
* ''Noncompetitive inhibitors:'' [[Trilostane]]
−
    | list2 = {{Navbox subgroup
 
−
    | groupstyle = text-align:center;
 
  
−
      | group1 = Agonists
+
  }}
−
      | list1 =
+
 
 +
  | group2 = {{abbrlink|GPER|G protein-coupled estrogen receptor}}
 +
  | list2 = {{Navbox|subgroup
 +
  | groupstyle = text-align:center
 +
  | groupwidth = 6em;
 +
 
 +
    | group1 = Agonists
 +
    | list1 =
 +
* [[2-Methoxyestradiol]]
 
* [[7β-Hydroxyepiandrosterone]]
 
* [[7β-Hydroxyepiandrosterone]]
 
* [[Afimoxifene|Afimoxifene (4-hydroxytamoxifen)]]
 
* [[Afimoxifene|Afimoxifene (4-hydroxytamoxifen)]]
 +
* [[Aldosterone]]
 
* [[Atrazine]]
 
* [[Atrazine]]
 
* [[Bisphenol A]]
 
* [[Bisphenol A]]
 
* [[Daidzein]]
 
* [[Daidzein]]
 
* [[DDT]] ([[p,p'-DDT]], [[o',p'-DDE]])
 
* [[DDT]] ([[p,p'-DDT]], [[o',p'-DDE]])
 +
* [[Diarylpropionitrile]]
 
* [[Equol]]
 
* [[Equol]]
 
* [[Estradiol]]
 
* [[Estradiol]]
−
* [[Fulvestrant|Fulvestrant (ICI-182,780)]]
+
* [[Ethinylestradiol]]
 +
* [[Fulvestrant|Fulvestrant (ICI-182780)]]
 
* [[G-1 (drug)|G-1]]
 
* [[G-1 (drug)|G-1]]
 
* [[Genistein]]
 
* [[Genistein]]
Line 246: Line 354:
 
* [[Nonylphenol]]
 
* [[Nonylphenol]]
 
* [[Oleuropein]]
 
* [[Oleuropein]]
−
* [[Polychlorinated biphenyl|PCB]] ([[2,2',5'-PCB-4-OH]])
+
* [[Polychlorinated biphenyl|PCB]]s ([[2,2',5'-PCB-4-OH]])
 
* [[Propylpyrazoletriol]]
 
* [[Propylpyrazoletriol]]
 
* [[Quercetin]]
 
* [[Quercetin]]
 
* [[Raloxifene]]
 
* [[Raloxifene]]
 
* [[Resveratrol]]
 
* [[Resveratrol]]
 +
* [[STX (drug)|STX]]
 
* [[Tamoxifen]]
 
* [[Tamoxifen]]
 
* [[Tectoridin]]
 
* [[Tectoridin]]
−
* [[Zearalenone]]
 
  
−
      | group2 = Antagonists
+
    | group2 = Antagonists
−
      | list2 =
+
    | list2 =
 +
* [[CCL18]]
 
* [[Estriol]]
 
* [[Estriol]]
 
* [[G-15 (drug)|G-15]]
 
* [[G-15 (drug)|G-15]]
Line 262: Line 371:
 
* [[MIBE]]
 
* [[MIBE]]
  
−
     }}
+
     | group3 = Unknown
 +
    | list3 =
 +
* [[Diethylstilbestrol]]
 +
* [[Zearalenone]]
 +
 
 
   }}
 
   }}
  
−
   | group2 = [[Enzyme]]
+
<!--
−
   | list2  = {{Navbox subgroup
+
   | group3 = {{abbrlink|ER-X|Estrogen receptor X}}
 +
   | list3 = {{Navbox|subgroup
 +
  | groupstyle = text-align:center
 +
  | groupwidth = 6em;
  
−
     | group1 = [[Enzyme modulator|Modulators]]
+
     | group1 = Agonists
 
     | list1 =
 
     | list1 =
−
* See [[Template:Steroid hormone metabolism modulators|here]] instead (modulators of [[cholesterol side-chain cleavage enzyme|20,22-desmolase]], [[CYP17A1|17α-hydroxylase/17,20-lyase]], [[3β-Hydroxysteroid dehydrogenase|3β-HSD]], [[17β-Hydroxysteroid dehydrogenase|17β-HSD]], [[5α-reductase]], [[aromatase]], and [[CYP27A1|27-hydroxylase]]).
+
* [[Alfatradiol|17α-Estradiol (alfatradiol)]]
 +
* [[Estradiol]]
 +
 
 +
    | group2 = Antagonists
 +
    | list2 =
  
−
    }}
+
  }}
  
−
   | group3 = Others
+
   | group4 = {{abbrlink|G<sub>q</sub>-mER|Gq-coupled membrane estrogen receptor}}
−
   | list3 = {{Navbox subgroup
+
   | list4 = {{Navbox|subgroup
−
   | groupstyle = text-align:center;
+
   | groupstyle = text-align:center
 +
  | groupwidth = 6em;
  
−
     | group1 = Precursors
+
     | group1 = Agonists
 
     | list1 =
 
     | list1 =
−
* [[Cholesterol]]
+
* [[Estradiol]]
−
* [[22R-Hydroxycholesterol|22''R''-Hydroxycholesterol]]
+
* [[STX (drug)|STX]]
−
* [[20α,22R-Dihydroxycholesterol|20α,22''R''-Dihydroxycholesterol]]
 
−
* [[Pregnenolone]]
 
−
* [[Pregnenolone sulfate]]
 
−
* [[17-Hydroxypregnenolone]]
 
−
* [[Progesterone]]
 
−
* [[17-Hydroxyprogesterone]]
 
−
* [[11-Deoxycortisol|11-Deoxycortisol (cortodoxone)]]
 
−
* [[Dehydroepiandrosterone|DHEA]]
 
−
* [[Dehydroepiandrosterone sulfate|DHEA sulfate]]
 
−
* [[16-Hydroxydehydroepiandrosterone sulfate|16-Hydroxy-DHEA sulfate]]
 
−
* [[Δ5-Androstenediol|Δ<sup>5</sup>-Androstenediol]]
 
−
* [[Δ4-Androstenedione|Δ<sup>4</sup>-Androstenedione]]
 
−
* [[16-Hydroxyandrostenedione]]
 
−
* [[Testosterone]]
 
  
−
  | group2 = Indirect
+
    | group2 = Antagonists
−
  | list2 =
+
    | list2 =
−
* [[Antigonadotropin]]s (e.g., [[androgen]]s, [[estrogen]]s, [[progestogen]]s, [[prolactin]])
+
* [[Fulvestrant|Fulvestrant (ICI-182780)]]
−
* [[Calcitriol]] ([[vitamin D]])
 
−
* [[Gonadotropin-releasing hormone agonist|GnRH agonists]] (e,g, [[gonadotropin-releasing hormone|GnRH]], [[leuprorelin]])
 
−
* [[Gonadotropin-releasing hormone antagonist|GnRH antagonists]] (e.g., [[cetrorelix]])
 
−
* [[Gonadotropin]]s (e.g., [[follicle-stimulating hormone|FSH]], [[human chorionic gonadotropin|hCG]], [[luteinizing hormone|LH]])
 
−
* [[Kisspeptin]]
 
−
* [[Plasma protein]]s ([[Androgen-binding protein|ABP]], [[serum albumin|albumin]], [[Sex hormone-binding globulin|SHBG]])
 
  
−
    }}
+
  }}
 +
-->
  
−
   | below = '''''See also:''' [[Template:Androgenics|Androgenics]] • [[Template:Glucocorticoid signaling|Glucocorticoids]] • [[Template:Mineralocorticoid signaling|Mineralocorticoids]] • [[Template:Progestogenics|Progestogenics]]''
+
   | below =  
 +
;See also
 +
: [[Template:Receptor modulators|Receptor/signaling modulators]]  
 +
: [[Template:Estrogens and antiestrogens|Estrogens and antiestrogens]]  
 +
: [[Template:Androgen receptor modulators|Androgen receptor modulators]]  
 +
: [[Template:Progesterone receptor modulators|Progesterone receptor modulators]]
 +
: [[List of steroidal estrogens|List of estrogens]]
  
−
}}<noinclude>
+
}}
 +
<noinclude>
 
{{collapsible option}}
 
{{collapsible option}}
 
[[Category:Drug templates by receptor, channel, or pump]]
 
[[Category:Drug templates by receptor, channel, or pump]]
 
[[Category:Estrogens]]
 
[[Category:Estrogens]]
 
</noinclude>
 
</noinclude>

Latest revision as of 18:59, 30 July 2020

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