Difference between revisions of "Template:Anticholinergics"

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blackwiki>Sir Pinade
(nicotine -> depolarizing agent + other molecules)
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   | group1 = [[Ganglionic blocker|Ganglionic]]
 
   | group1 = [[Ganglionic blocker|Ganglionic]]
   |  list1 = ''nondepolarizing'' ([[Mecamylamine]], [[Trimetaphan camsilate|Trimetaphan]], [[Hexamethonium]]){{·}} [[Nicotine|Nicotine (high doses)]]<BR>''note: in [[Parasympathetic nervous system|PNS]], ganglionic blocker can have direct '''antinicotinic''' action at [[Preganglionic fibers|preganglionic]] terminal, but simulate indirect '''antimuscarinic''' activities at [[Postganglionic fibers|postganglionic]] terminal
+
   |  list1 = ''nondepolarizing:'' [[Hexamethonium]], [[Mecamylamine]], [[Pentolinium]], [[Trimetaphan camsilate|Trimetaphan]]
 +
 
 +
''depolarizing:'' [[Nicotine|Nicotine (high doses)]] <BR>''note: in [[Parasympathetic nervous system|PNS]], ganglionic blocker can have direct '''antinicotinic''' action at [[Preganglionic fibers|preganglionic]] terminal, but simulate indirect '''antimuscarinic''' activities at [[Postganglionic fibers|postganglionic]] terminal
  
 
   | group2 = [[Neuromuscular blocker|Neuromuscular]]
 
   | group2 = [[Neuromuscular blocker|Neuromuscular]]
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|  list2 = ''nonpolar/tertiary/[[Blood-brain barrier|CNS]]:'' [[Atropine]]{{·}} [[Scopolamine]]{{·}} [[Hyoscyamine]]{{·}} ''[[antiparkinson drug]]s'' ([[Benzatropine]], [[Trihexyphenidyl]], [[Biperiden]])
 
|  list2 = ''nonpolar/tertiary/[[Blood-brain barrier|CNS]]:'' [[Atropine]]{{·}} [[Scopolamine]]{{·}} [[Hyoscyamine]]{{·}} ''[[antiparkinson drug]]s'' ([[Benzatropine]], [[Trihexyphenidyl]], [[Biperiden]])
  
''polar/quarternary/non-CNS:'' [[Glycopyrrolate]]{{·}} [[Ipratropium]]{{·}} [[Muscarinic acetylcholine receptor M1|M1]] ([[Pirenzepine]]){{·}} [[Muscarinic acetylcholine receptor M3|M3]] ([[Tiotropium]], [[Darifenacin]], [[Vedaclidine]])
+
''polar/quarternary/non-CNS:'' [[Glycopyrrolate]]{{·}} [[Ipratropium]]{{·}} [[Muscarinic acetylcholine receptor M1|M1]] ([[Pirenzepine]], [[Telenzepine]]){{·}} [[Muscarinic acetylcholine receptor M3|M3]] ([[Tiotropium]], [[Darifenacin]], [[Vedaclidine]])
  
 
''unsorted:'' [[Tropicamide]]{{·}} [[Cyclopentolate]]{{·}} [[Dicycloverine]]{{·}} [[Tolterodine]]{{·}} [[Oxybutynin]]{{·}} [[Homatropine]] {{·}} [[Orphenadrine]]{{·}} [[Diphenhydramine]]{{·}} Other ethanolamine class first-generation [[antihistamines]]
 
''unsorted:'' [[Tropicamide]]{{·}} [[Cyclopentolate]]{{·}} [[Dicycloverine]]{{·}} [[Tolterodine]]{{·}} [[Oxybutynin]]{{·}} [[Homatropine]] {{·}} [[Orphenadrine]]{{·}} [[Diphenhydramine]]{{·}} Other ethanolamine class first-generation [[antihistamines]]

Revision as of 18:51, 23 April 2009