Difference between revisions of "Template:Anticholinergics"
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blackwiki>Sir Pinade (nicotine -> depolarizing agent + other molecules) |
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| group1 = [[Ganglionic blocker|Ganglionic]] | | group1 = [[Ganglionic blocker|Ganglionic]] | ||
| − | | list1 = ''nondepolarizing'' | + | | list1 = ''nondepolarizing:'' [[Hexamethonium]], [[Mecamylamine]], [[Pentolinium]], [[Trimetaphan camsilate|Trimetaphan]] |
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| + | ''depolarizing:'' [[Nicotine|Nicotine (high doses)]] <BR>''note: in [[Parasympathetic nervous system|PNS]], ganglionic blocker can have direct '''antinicotinic''' action at [[Preganglionic fibers|preganglionic]] terminal, but simulate indirect '''antimuscarinic''' activities at [[Postganglionic fibers|postganglionic]] terminal | ||
| group2 = [[Neuromuscular blocker|Neuromuscular]] | | group2 = [[Neuromuscular blocker|Neuromuscular]] | ||
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| list2 = ''nonpolar/tertiary/[[Blood-brain barrier|CNS]]:'' [[Atropine]]{{·}} [[Scopolamine]]{{·}} [[Hyoscyamine]]{{·}} ''[[antiparkinson drug]]s'' ([[Benzatropine]], [[Trihexyphenidyl]], [[Biperiden]]) | | list2 = ''nonpolar/tertiary/[[Blood-brain barrier|CNS]]:'' [[Atropine]]{{·}} [[Scopolamine]]{{·}} [[Hyoscyamine]]{{·}} ''[[antiparkinson drug]]s'' ([[Benzatropine]], [[Trihexyphenidyl]], [[Biperiden]]) | ||
| − | ''polar/quarternary/non-CNS:'' [[Glycopyrrolate]]{{·}} [[Ipratropium]]{{·}} [[Muscarinic acetylcholine receptor M1|M1]] ([[Pirenzepine]]){{·}} [[Muscarinic acetylcholine receptor M3|M3]] ([[Tiotropium]], [[Darifenacin]], [[Vedaclidine]]) | + | ''polar/quarternary/non-CNS:'' [[Glycopyrrolate]]{{·}} [[Ipratropium]]{{·}} [[Muscarinic acetylcholine receptor M1|M1]] ([[Pirenzepine]], [[Telenzepine]]){{·}} [[Muscarinic acetylcholine receptor M3|M3]] ([[Tiotropium]], [[Darifenacin]], [[Vedaclidine]]) |
''unsorted:'' [[Tropicamide]]{{·}} [[Cyclopentolate]]{{·}} [[Dicycloverine]]{{·}} [[Tolterodine]]{{·}} [[Oxybutynin]]{{·}} [[Homatropine]] {{·}} [[Orphenadrine]]{{·}} [[Diphenhydramine]]{{·}} Other ethanolamine class first-generation [[antihistamines]] | ''unsorted:'' [[Tropicamide]]{{·}} [[Cyclopentolate]]{{·}} [[Dicycloverine]]{{·}} [[Tolterodine]]{{·}} [[Oxybutynin]]{{·}} [[Homatropine]] {{·}} [[Orphenadrine]]{{·}} [[Diphenhydramine]]{{·}} Other ethanolamine class first-generation [[antihistamines]] | ||