Template:Antiandrogens marketed for clinical or veterinary use
Revision as of 11:50, 27 March 2019 by 84.250.17.211 (talk) (Table footer: Use tfoot for notes/references)
| Generic name | Class | Type | Brand name(s) | Route(s) | Launch | Status | Hitsa |
|---|---|---|---|---|---|---|---|
| Abiraterone acetate | Steroidal | Androgen synthesis inhibitor | Zytiga | Oral | 2011 | Available | 523,000 |
| Allylestrenol | Steroidal | Progestin | Gestanin, Perselin | Oral | 1961 | Availableb | 61,800 |
| Aminoglutethimide | Nonsteroidal | Androgen synthesis inhibitor | Cytadren, Orimeten | Oral | 1960 | Availableb | 222,000 |
| Apalutamide | Nonsteroidal | AR antagonist | Erleada | Oral | 2018 | Available | 50,400 |
| Bicalutamide | Nonsteroidal | AR antagonist | Casodex | Oral | 1995 | Available | 754,000 |
| Chlormadinone acetate | Steroidal | Progestin; AR antagonist | Belara, Prostal | Oral | 1965 | Available | 220,000 |
| Cyproterone acetate | Steroidal | Progestin; AR antagonist | Androcur, Diane | Oral, IM | 1973 | Available | 461,000 |
| Delmadinone acetate | Steroidal | Progestin; AR antagonist | Tardak | Veterinary | 1972 | Veterinary | 42,600 |
| Enzalutamide | Nonsteroidal | AR antagonist | Xtandi | Oral | 2012 | Available | 328,000 |
| Flutamide | Nonsteroidal | AR antagonist | Eulexin | Oral | 1983 | Available | 712,000 |
| Gestonorone caproate | Steroidal | Progestin | Depostat, Primostat | IM | 1973 | Availableb | 119,000 |
| Hydroxyprogesterone caproate | Steroidal | Progestin | Delalutin, Proluton | IM | 1954 | Available | 108,000 |
| Ketoconazole | Nonsteroidal | Androgen synthesis inhibitor | Nizoral, others | Oral, topical | 1977 | Available | 3,650,000 |
| Medroxyprogesterone acetate | Steroidal | Progestin | Provera, Depo-Provera | Oral, IM, SC | 1958 | Available | 1,250,000 |
| Megestrol acetate | Steroidal | Progestin; AR antagonist | Megace | Oral | 1963 | Available | 253,000 |
| Nilutamide | Nonsteroidal | AR antagonist | Anandron, Nilandron | Oral | 1987 | Available | 132,000 |
| Osaterone acetate | Steroidal | Progestin; AR antagonist | Ypozane | Veterinary | 2007 | Veterinary | 87,600 |
| Oxendolone | Steroidal | Progestin; AR antagonist | Prostetin, Roxenone | IM | 1981 | Availableb | 36,100 |
| Spironolactone | Steroidal | AR antagonist | Aldactone | Oral, topical | 1959 | Available | 3,010,000 |
| Topilutamide | Nonsteroidal | AR antagonist | Eucapil | Topical | 2003 | Availableb | 36,300 |
| Footnotes: a = Hits = Google Search hits (as of February 2018). b = Availability limited / mostly discontinued. Class: Steroidal = Steroidal antiandrogen. Nonsteroidal = Nonsteroidal antiandrogen. Sources: See individual articles. | |||||||