Template:Anticholinergics
Revision as of 17:30, 3 October 2008 by blackwiki>Arcadian (Nicotine)
| Nicotinic antagonists | |
|---|---|
| Muscarinic antagonists | nonpolar/tertiary/CNS: Atropine · Scopolamine
polar/quarternary/non-CNS: Pirenzepine unsorted: Ipratropium · Tropicamide · Cyclopentolate · Benzatropine · Dicycloverine · Tolterodine · Oxybutynin · Biperiden · Trihexyphenidyl · Homatropine · M1 (Pirenzepine) · M3 (Tiotropium, Darifenacin) |
| Presynaptic | acetylcholine synthesis (Hemicholinium-3) · acetylcholine release (Botulinum toxin) |
| Other | acetylcholinesterase reactivators (Pralidoxime, Obidoxime) |
note: in PNS, ganglionic blocker can have direct antinicotinic action at preganglionic terminal, but simulate indirect antimuscarinic activities at postganglionic terminal | |