Template:Anticholinergics
Revision as of 12:59, 4 October 2008 by blackwiki>Arcadian (grouping)
| Nicotinic antagonists | |
|---|---|
| Muscarinic antagonists | nonpolar/tertiary/CNS: Atropine · Scopolamine
polar/quarternary/non-CNS: M1 (Pirenzepine) · M3 (Tiotropium, Darifenacin) unsorted: Ipratropium · Tropicamide · Cyclopentolate · Dicycloverine · Tolterodine · Oxybutynin · Homatropine · antiparkinson drugs (Benzatropine, Trihexyphenidyl, Biperiden) |
| Presynaptic | acetylcholine synthesis inhibitor (Hemicholinium-3) · acetylcholine release inhibitor (Botulinum toxin) - acetylcholine release stimulator (Alpha-latrotoxin) |
| Other | acetylcholinesterase reactivators (Pralidoxime, Obidoxime) |
note: in PNS, ganglionic blocker can have direct antinicotinic action at preganglionic terminal, but simulate indirect antimuscarinic activities at postganglionic terminal | |