Template:Major estrogens marketed for clinical or veterinary use

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Major Template:No selflinks marketed for clinical or veterinary use

Generic name Class Brand name(s) Route(s) Launch Status Hitsa
Chlorotrianisene Nonsteroidal Tace, others Oral 1952 Discontinued 473,000
Conjugated estriol Steroidal; Ester Emmenin, Progynon Oral, others 1930 Discontinued –
Conjugated estrogens Steroidal; Equine; Ester Premarin Oral, others 1941 Available 2,800,000
Dienestrol Nonsteroidal Numerous Oral 1947 Availableb 527,000
Diethylstilbestrol Nonsteroidal Stilbestrol, others Oral, others 1939 Availableb 560,000
Diethylstilbestrol dipropionate Nonsteroidal; Ester Numerous IM 1940s Discontinued 2,790
Esterified estrogens Steroidal; Equine; Ester Estratab Oral 1970 Available 113,000
Estetrol Steroidal Donesta, Estelle Oral Phase III Experimental 24,000
Estradiol Steroidal Estrace, numerous others Many 1935 Available 9,720,000
Estradiol acetate Steroidal; Ester Femtrace, Femring, Menoring Oral, vaginal 2001 Available 50,900
Estradiol benzoate Steroidal; Ester Progynon B IM 1933 Available 177,000
Estradiol cypionate Steroidal; Ester Depo-Estradiol IM 1952 Available 75,900
Estradiol dipropionate Steroidal; Ester Agofollin, Di-Ovocyclin, Progynon DP IM 1939 Discontinued 12,400
Estradiol enanthate Steroidal; Ester Deladroxate, Perlutan, Topasel IM 1970s Available 44,600
Estradiol undecylate Steroidal; Ester Progynon Depot 100 IM 1956 Discontinued 8,250
Estradiol valerate Steroidal; Ester Progynova, Progynon Depot, Delestrogen Oral, IM 1954 Available 2,200,000
Estramustine phosphate Steroidal; Ester; Cytostatic Emcyt, Estracyt Oral 1970s Available 237,000
Estriol Steroidal Theelol, Ovestin Oral, vaginal 1930 Available 8,930,000
Estrogenic substances Steroidal Amniotin, others Oral, others 1929 Discontinued –
Estrone Steroidal Theelin, others IM 1929 Discontinued 850,000
Estropipate Steroidal; Ester Ogen Oral 1968 Availableb 214,000
Ethinylestradiol Steroidal; Alkyl Estinyl, numerous others Oral, others 1943 Available 1,780,000
Ethinylestradiol sulfonate Steroidal; Alkyl; Ester Deposiston, Turisteron Oral 1978 Discontinued 10,900
Fosfestrol Nonsteroidal; Ester Honvan, others IM 1947 Availableb 115,000
Hexestrol Nonsteroidal Synestrol, others Oral, others 1940s Availableb 171,000
Mestranol Steroidal; Alkyl; Ether Numerous Oral 1957 Availableb 169,000
Methallenestril Nonsteroidal; Ether Vallestril Oral 1950s Discontinued 35,300
Methylestradiol Steroidal; Alkyl Ginecosid, others Oral 1955 Availableb 10,500
Moxestrol Steroidal; Alkyl Surestryl Oral 1970s Discontinued 9,510
Polyestradiol phosphate Steroidal; Ester; Polymer Estradurin IM 1957 Availableb 124,000
Polyestriol phosphate Steroidal; Ester; Polymer Gynäsan, Klimadurin, Triodurin IM 1968 Discontinued 2,040
Prasterone (DHEA) Steroidal; Prohormone Numerous Many 1970s Available 11,600,000
Quinestrol Steroidal; Alkyl; Ether Estrovis Oral 1960s Discontinued 23,800
Zeranol Nonsteroidal Ralgro, others Veterinary 1970s Veterinary 91,800
Footnotes: a = Hits = Google Search hits (as of February 2018). b = Availability limited / mostly discontinued. Class: Steroidal = Steroidal estrogen. Nonsteroidal = Nonsteroidal estrogen. Alkyl = 17α-Alkylated. Cytostatic = Chemotherapeutic agent. Sources: See individual articles.